| 产品描述: | Aminohexylgeldanamycin (AHGDM), a Geldanamycin derivative, is a potent HSP90 inhibitor. Aminohexylgeldanamycin shows antiangiogenic and antitumor activities. |
| 靶点: |
HSP90 |
| 体内研究: |
HPMA copolymer-aminohexylgeldanamycin conjugates 在前列腺癌中靶向细胞表面表达的 GRP78。 |
| 参考文献: |
1. Greish K, et al. Anticancer and antiangiogenic activity of HPMA copolymer-aminohexylgeldanamycin-RGDfK conjugates for prostate cancer therapy. J Control Release. 2011;151(3):263-270. |
| 保存条件: |
-80°C 6个月; -20°C 1个月,避光 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.551 ml |
7.754 ml |
15.509 ml |
| 5 mM |
0.31 ml |
1.551 ml |
3.102 ml |
| 10 mM |
0.155 ml |
0.775 ml |
1.551 ml |
| 50 mM |
0.031 ml |
0.155 ml |
0.31 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |