| 产品描述: | DPP-IV-IN-1 is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV), a highly specific serine protease, with an IC50 of 4.6 nM. |
| 靶点: |
DPP-4 |
| 体外研究: |
DPP-IV-IN-1 (0.1 and 0.3 mg/kg, p.o.) reduces the increase in plasma glucose beginning 30 min after glucose loading, and significantly suppresses hyperglycemia at the dose of 0.3 mg/kg in a rat model of obesity and impaired glucose tolerance. The effect is based on its inhibitory effect on plasma DPP-IV activity[1]. |
| 保存条件: |
-80°C 6个月;-20°C 1个月 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
4.11 ml |
20.552 ml |
41.105 ml |
| 5 mM |
0.822 ml |
4.11 ml |
8.221 ml |
| 10 mM |
0.411 ml |
2.055 ml |
4.11 ml |
| 50 mM |
0.082 ml |
0.411 ml |
0.822 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |