Misetionamide is an orally oxathiazin-like compound. Misetionamide is a glyceraldehyde-3-phosphate dehydrogenase (GAPDH) inhibitor with antineoplastic activity. Misetionamide can be used for the research of cancer.
体内研究:
Misetionamide (OTD) (0-2000 μM; 0-72 h) induces cell death in TNBC cells. Misetionamide (OTD) (0-2000 μM; 12 h) inhibits TNBC cells proliferation. Misetionamide (OTD) (0-1000 μM; 18 h) induces necrosis and apoptosis in TNBC cells. Misetionamide (OTD) (250-1000 μM; 18 h) induces cell death by a ROS-dependent mechanism in TNBC cells.