| 产品描述: | Curcumin 5-8 (CUR5-8) is a potent and orally active naturally active curcumin (CUR) analog. Curcumin 5-8 inhibits lipid droplet formation. Curcumin 5-8 increases autophagy and inhibits Apoptosis. Curcumin 5-8 improves insulin resistance and insulin sensitivity. |
| 体外研究: |
Curcumin 5-8 (100 mg/kg; diet; daily for 13 weeks) 改善 HFD (高脂肪饮食) 诱导的肥胖小鼠的胰岛素抵抗和肝脂肪变性[1]。 |
| 体内研究: |
Curcumin 5-8 (20 µM; 24 h) 降低 AML12 细胞中 PA (palmitic acid ) 诱导的 SREBP1 表达水平并增加 Bcl2/BAX 表达。 |
| 保存条件: |
-80°C 6个月;-20°C 1个月 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.946 ml |
14.732 ml |
29.465 ml |
| 5 mM |
0.589 ml |
2.946 ml |
5.893 ml |
| 10 mM |
0.295 ml |
1.473 ml |
2.946 ml |
| 50 mM |
0.059 ml |
0.295 ml |
0.589 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |