| 产品描述: | Crisnatol (BWA770U) is an orally active and anticancer agent, and a member of the arylmethylaminopropanediol class of DNA intercalators. Crisnatol shows in vitro cytotoxicity against human breast cancer cells, but not normal human skin fibroblasts. |
| 体外研究: |
Crisnatol (25 mg/kg; p.o.; single dose) 显示出口服活性,并通过放射自显影显示大鼠粪便提取物的稳定代谢物谱[2]。 |
| 体内研究: |
Crisnatol (1.3 μg/mL; 24-72 h) 抑制 HepG2 细胞的复制,使细胞活力降低 35%。 |
| 保存条件: |
-80°C 12个月; -20°C 6个月,干燥, 避光 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.895 ml |
14.475 ml |
28.949 ml |
| 5 mM |
0.579 ml |
2.895 ml |
5.79 ml |
| 10 mM |
0.289 ml |
1.447 ml |
2.895 ml |
| 50 mM |
0.058 ml |
0.289 ml |
0.579 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |