(R)-lunresertib is a membrane-associated tyrosine and threonine-specific cdc2-inhibitory kinase (Myt1) (Gene name PKMYT1) inhibitor, with IC50 of 1360 nM. (R)-lunresertib can be used in the study of Myt1-mediated cancers.
靶点:
PKMYT1
参考文献:
1. Daniel Durocher, et al. Methods of using myt1 inhibitors. Pantent WO2021195782A1.